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Arisa Masuda
Arisa Masuda
International University, Cambodia
Chemistry
Biochemistry
Farnesoid X receptor
Structure–activity relationship
Plasmin Inhibitors
4
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14
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Design and identification of a new farnesoid X receptor (FXR) partial agonist by computational structure-activity analysis: Ligand-induced H8 helix fluctuation in the ligand-binding domain of FXR may lead to partial agonism.
2021
Bioorganic & Medicinal Chemistry Letters
Keigo Gohda
Yusuke Iguchi
Arisa Masuda
Ko Fujimori
Yukiko Yamashita
Naoki Teno
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N1-Substituted benzimidazole scaffold for farnesoid X receptor (FXR) agonists accompanying prominent selectivity against vitamin D receptor (VDR)
2020
Bioorganic & Medicinal Chemistry
Arisa Masuda
Keigo Gohda
Yusuke Iguchi
Ko Fujimori
Yukiko Yamashita
Keisuke Oda
Mizuho Une
Naoki Teno
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Identification of potent farnesoid X receptor (FXR) antagonist showing favorable PK profile and distribution toward target tissues: Comprehensive understanding of structure-activity relationship of FXR antagonists
2019
Bioorganic & Medicinal Chemistry
Naoki Teno
Yukiko Yamashita
Arisa Masuda
Yusuke Iguchi
Keisuke Oda
Ko Fujimori
Takie Hiramoto
Tomoko Nishimaki-Mogami
Mizuho Une
Keigo Gohda
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Novel type of plasmin inhibitors: Providing insight into P4 moiety and alternative scaffold to pyrrolopyrimidine
2015
Bioorganic & Medicinal Chemistry
Naoki Teno
Keigo Gohda
Keiko Wanaka
Yuko Tsuda
Maiko Akagawa
Eriko Akiduki
Mitsuhito Araki
Arisa Masuda
Tadamune Otsubo
Yukiko Yamashita
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Citations (8)
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