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Xilin Lyu
Xilin Lyu
Chinese Academy of Sciences
Chemistry
Biochemistry
Kinase
Drug discovery
Growth inhibition
5
Papers
32
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Recent Progress and Clinical Development of Inhibitors that Block MDM4/p53 Protein-Protein Interactions.
2021
Journal of Medicinal Chemistry
Shiyan Zhang
Jianfeng Lou
Yafang Li
Feilong Zhou
Ziqin Yan
Xilin Lyu
Yujun Zhao
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Synthesis and Bioactivity Studies of Covalent Inhibitors Derived from (-)-Chaetominine
2021
Journal of Molecular Structure
Xian Zhou
Xuexin Feng
Dachi Wang
Chen Deheng
Gaoxing Wu
Ziqin Yan
Xilin Lyu
Huan Wang
Jin-Ming Yang
Yujun Zhao
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Discovery of a potent and selective NF-κB-inducing kinase (NIK) inhibitor that has anti-inflammatory effects in vitro and in vivo
2020
Journal of Medicinal Chemistry
Zhiqiang Li
Xinzhi Li
Mingbo Su
Li-Xin Gao
Yubo Zhou
Bingchuan Yuan
Xilin Lyu
Ziqin Yan
Chujiao Hu
Hao Zhang
Cheng Luo
Zheng Chen
Jia Li
Yujun Zhao
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Discovery of a 2-pyridinyl urea-containing compound YD57 as a potent inhibitor of apoptosis signal-regulating kinase 1 (ASK1)
2020
European Journal of Medicinal Chemistry
Shiyan Zhang
Chaoying Huang
Xilin Lyu
Peipei Wang
Yi Zang
Zengtao Wang
Huan Wang
Jia Li
Yujun Zhao
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Discovery, structural insight, and bioactivities of BY27 as a selective inhibitor of the second bromodomains of BET proteins
2019
European Journal of Medicinal Chemistry
Deheng Chen
Tian Lu
Ziqin Yan
Wenchao Lu
Feilong Zhou
Xilin Lyu
Biling Xu
Hualiang Jiang
Kaixian Chen
Cheng Luo
Yujun Zhao
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