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Lijie Zhao
Lijie Zhao
University of Michigan
Chemistry
Cancer research
Androgen receptor
Apoptosis
Cell culture
5
Papers
75
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Discovery of ARD-2585 as an Exceptionally Potent and Orally Active PROTAC Degrader of Androgen Receptor for the Treatment of Advanced Prostate Cancer.
2021
Journal of Medicinal Chemistry
Weiguo Xiang
Lijie Zhao
Xin Han
Chong Qin
Bukeyan Miao
Donna McEachern
Yu Wang
Hoda Metwally
Paul D. Kirchhoff
Lu Wang
Aleksas Matvekas
Miao He
Bo Wen
Duxin Sun
Shaomeng Wang
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Strategies toward Discovery of Potent and Orally Bioavailable Proteolysis Targeting Chimera Degraders of Androgen Receptor for the Treatment of Prostate Cancer.
2021
Journal of Medicinal Chemistry
Xin Han
Lijie Zhao
Weiguo Xiang
Chong Qin
Bukeyan Miao
Donna McEachern
Yu Wang
Hoda Metwally
Lu Wang
Aleksas Matvekas
Bo Wen
Duxin Sun
Shaomeng Wang
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A highly potent PROTAC androgen receptor (AR) degrader ARD-61 effectively inhibits AR-positive breast cancer cell growth in vitro and tumor growth in vivo.
2020
Neoplasia
Lijie Zhao
Xin Han
Jianfeng Lu
Donna McEachern
Shaomeng Wang
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Citations (13)
Discovery of Highly Potent and Efficient PROTAC Degraders of Androgen Receptor (AR) by Employing Weak Binding Affinity VHL E3 Ligase Ligands
2019
Journal of Medicinal Chemistry
Xin Han
Lijie Zhao
Weiguo Xiang
Chong Qin
Bukeyan Miao
Tianfeng Xu
Mi Wang
Chao Yie Yang
Krishnapriya Chinnaswamy
Jeanne A. Stuckey
Shaomeng Wang
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Citations (47)
Discovery of [1,2,4]triazolo[1,5-a]pyrimidine derivatives as new bromodomain-containing protein 4 (BRD4) inhibitors
2019
Chinese Chemical Letters
Shuai Wang
Dan-Dan Shen
Lijie Zhao
Xiao-Han Yuan
Jialing Cheng
Bin Yu
Yi-Chao Zheng
Hong-Min Liu
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Citations (15)
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