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Takie Hiramoto
Takie Hiramoto
International University, Cambodia
Biochemistry
Farnesoid X receptor
Pharmacology
Antagonist
In vivo
2
Papers
11
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Identification of potent farnesoid X receptor (FXR) antagonist showing favorable PK profile and distribution toward target tissues: Comprehensive understanding of structure-activity relationship of FXR antagonists
2019
Bioorganic & Medicinal Chemistry
Naoki Teno
Yukiko Yamashita
Arisa Masuda
Yusuke Iguchi
Keisuke Oda
Ko Fujimori
Takie Hiramoto
Tomoko Nishimaki-Mogami
Mizuho Une
Keigo Gohda
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Citations (3)
Nonacidic Chemotype Possessing N-Acylated Piperidine Moiety as Potent Farnesoid X Receptor (FXR) Antagonists
2018
ACS Medicinal Chemistry Letters
Naoki Teno
Yukiko Yamashita
Yusuke Iguchi
Ko Fujimori
Mizuho Une
Tomoko Nishimaki-Mogami
Takie Hiramoto
Keigo Gohda
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Citations (8)
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