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Melissa D. Chengalroyen
Melissa D. Chengalroyen
University of Cape Town
Mycobacterium tuberculosis
Chemistry
Biochemistry
Prodrug
Isoniazid
2
Papers
4
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0
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DNA-dependent binding of nargenicin to DnaE1 inhibits replication in Mycobacterium tuberculosis
2021
bioRxiv
Melissa D. Chengalroyen
Mandy K. Mason
Alessandro Borsellini
Raffaella Tassoni
Garth L. Abrahams
Sasha L. Lynch
Yong-Mo Ahn
Jon Ambler
Katherine Young
Brendan M. Crowley
David B. Olsen
Digby F. Warner
Clifton E. Barry
Helena I. Boshoff
Meindert H. Lamers
Valerie Mizrahi
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Citations (1)
Biological Profiling Enables Rapid Mechanistic Classification of Phenotypic Screening Hits and Identification of KatG Activation-Dependent Pyridine Carboxamide Prodrugs With Activity Against Mycobacterium tuberculosis
2020
Frontiers in Cellular and Infection Microbiology
Melissa D. Chengalroyen
Audrey Jordaan
Ronnett Seldon
Thomas R. Ioerger
Scott G. Franzblau
Mohamed Nasr
Digby F. Warner
Valerie Mizrahi
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